SCHEMBL6452765

SCHEMBL6452765

CCOC(C(N)=O)c1c(F)ccc(OCC2CCCO2)c1F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.46
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
IRAK4 Q9NWZ3 4/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
PTGER1 P34995 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
MAPT P10636 1/20 0.38
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
HTR2A P28223 2/20 0.37
SLC6A4 P31645 2/20 0.37
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5042028 0.82 F10 (0.39) SCN9ATSHRKDM4EALDH1A1MEN1
SCHEMBL6452774 0.72 POLB (0.48) SCN9ATSHRL3MBTL1KDM4EALDH1A1
SCHEMBL30151904 0.71 SCN9A (0.53) SCN9ATSHRIRAK4KDM4EALDH1A1
SCHEMBL29397819 0.68 TSHR (0.43) SCN9ATSHRIRAK4KDM4EALDH1A1
SCHEMBL24337345 0.68 L3MBTL1 (0.42) SCN9ATSHRL3MBTL1KDM4EALDH1A1
SCHEMBL2814439 0.67 SCN9A (0.54) SCN9ATSHRKDM4EALDH1A1PTGER1
SCHEMBL2814888 0.67 SCN9A (0.54) SCN9ATSHRKDM4EALDH1A1PTGER1
SCHEMBL20090371 0.67 HTR2A (0.44) SCN9ATSHRL3MBTL1PTGER1MEN1
SCHEMBL12697009 0.67 ALDH1A1 (0.49) SCN9ATSHRKDM4EALDH1A1PTGER1
SCHEMBL12697089 0.67 ALDH1A1 (0.49) SCN9ATSHRKDM4EALDH1A1PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567498-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2005-08-31 EP disclosed
WO-2004048335-A2 MANDELIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2004-06-10 WO disclosed