SCHEMBL6454497

SCHEMBL6454497

O=C(O)c1ccc(CN2C(=O)c3cc(C#CCc4ccccc4)ccc3OS2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 11/20 0.50
SLC22A8 Q8TCC7 1/20 0.49
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
HPGD P15428 1/20 0.39
FFAR1 O14842 1/20 0.38
FFAR4 Q5NUL3 1/20 0.38
ENPP2 Q13822 1/20 0.36
PPARA Q07869 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6257299 0.83 MMP13 (0.44) MMP13SLC22A8KMT2AMEN1HPGD
SCHEMBL6240857 0.80 MMP13 (0.50) MMP13SLC22A8KMT2AMEN1HPGD
SCHEMBL6446546 0.79 MMP13 (0.49) MMP13SLC22A8KMT2AMEN1HPGD
SCHEMBL6767426 0.78 KMT2A (0.67) MMP13SLC22A8KMT2AMEN1HPGD
SCHEMBL6256775 0.73 MMP13 (0.42) MMP13SLC22A8HPGDENPP2
SCHEMBL6449268 0.71 MMP13 (0.51) MMP13SLC22A8KMT2AMEN1HPGD
SCHEMBL6450511 0.71 MMP13 (0.48) MMP13SLC22A8KMT2AMEN1HPGD
SCHEMBL6477654 0.69 MMP13 (0.52) MMP13SLC22A8
SCHEMBL6288447 0.69 MMP13 (0.58) MMP13SLC22A8FFAR1FFAR4
SCHEMBL6767433 0.69 MMP13 (0.46) MMP13SLC22A8KMT2AMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1536786-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2005-06-08 EP disclosed
EP-1434585-A1 ALKYNE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2004-07-07 EP disclosed
WO-2004006913-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed
WO-2003032999-A1 ALKYNE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2003-04-24 WO disclosed