SCHEMBL645480

SCHEMBL645480

COc1ccc2ccc[c]c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2A6 P11509 1/20 0.55
ACHE P22303 2/20 0.43
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 3/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 2/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HSD17B1 P14061 1/20 0.40
HSD17B2 P37059 1/20 0.40
NQO2 P16083 1/20 0.40
MAPK1 P28482 1/20 0.39
GSTP1 P09211 1/20 0.38
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA7 P43166 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2253346 0.87 CYP1A2 (0.55) CYP1A2CYP2A6ACHERAB9AKDM4E
SCHEMBL2254030 0.87 CYP1A2 (0.55) CYP1A2CYP2A6ACHERAB9AKDM4E
SCHEMBL152913 0.85 CYP1A2 (0.55) CYP1A2CYP2A6ACHERAB9AKDM4E
SCHEMBL2251601 0.80 NQO1 (0.43) CYP1A2KDM4EMEN1POLBKMT2A
SCHEMBL7197663 0.80 CYP1A2 (0.33) CYP1A2CYP2A6
SCHEMBL27961290 0.79 CYP1A2 (0.48) CYP1A2CYP2A6ACHERAB9AKDM4E
Magnesium Chloride Anhydrous SCHEMBL28811729 0.79 CYP1A2 (0.48) CYP1A2CYP2A6ACHERAB9AKDM4E
SCHEMBL5543057 0.77 GPR3 (0.40) CYP1A2RAB9AKDM4EKMT2ANPC1
SCHEMBL6583460 0.76 CYP1A2 (0.31) CYP1A2CYP2A6
SCHEMBL6048370 0.75 CA1 (0.43) CYP1A2CYP2A6ACHERAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 255 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117983302-A Catalyst containing ferrocene PNP ligand for ethylene selective tetramerization and preparation method and application thereof 华东理工大学 2024-05-07 CN claimed
CN-107353229-B A kind of preparation method of agomelatine intermediate body 许昌恒生制药有限公司 2019-04-30 CN claimed
CN-104230754-B A kind of synthetic method of (7-methoxy-1-naphthyl) acetonitrile ZHEJIANG UNIVERSITY OF SCIENCE AND TECHNOLOGY (CN) 2017-01-04 CN claimed
CN-104557591-B A kind of method preparing agomelatine acetyl diamines 扬子江药业集团四川海蓉药业有限公司 2016-09-07 CN claimed
CN-102234238-B Method for preparing 2-(7-methoxy-1-naphthyl) ethylamine industrially SHANGHAI INST PHARM INDUSTRY 2014-06-18 CN claimed
CN-103073441-A Novel method for compositing (7- methoxy-1-naphthyl) and application of method in compositing of agomelatine SHANGHAI RIGHT HAND MEDICAL TECHNOLOGY DEV CO LTD 2013-05-01 CN claimed
CN-101538201-B Preparation method of agomelatine midbody (7-methoxyl group-1-naphthyl) acetic ester SHANGHAI INST PHARM INDUSTRY 2013-03-06 CN claimed
CN-101792400-B Synthetic method for agomelatine UNIV EAST CHINA NORMAL 2013-01-30 CN claimed
US-6509426-B2 Dichloro(1,1'-dimethylsilylenebis(2-methyl-4-(4-methoxyphenyl) -4H-azulenyl))zirconium, for example; can produce polyolefin with high molecular weight and high melting point for extrusion or injection moldability JAPAN POLYCHEM CORPORATION (JP) 2003-01-21 US claimed
US-6127357-A N-((phenyl, benzodioxinyl or N-heteroarylpiperazinyl)alkyl)-N-(N-heteroaryl)substituted carboxamides JOHN WYETH & BROTHER, LTD. (GB) 2000-10-03 US claimed
EP-0512755-B1 Piperazine derivatives WYETH JOHN & BROTHER LTD (GB) 1994-12-14 EP claimed
EP-0354093-B1 Piperazine derivatives and process for their preparation SYNTHELABO (FR) 1993-12-22 EP claimed
EP-0512755-A2 Piperazine derivatives JOHN WYETH & BROTHER LIMITED (GB) 1992-11-11 EP claimed
EP-0354094-B1 INDOLONE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTICAL USE SYNTHELABO (FR) 1991-12-27 EP claimed
US-5010079-A Treatment of psychological disorders SYNTHELABO (FR) 1991-04-23 US claimed
US-4963680-A INTERMEDIATES FOR THERAPEUTIC DRUGS SYNTHELABO (FR) 1990-10-16 US claimed
JP-2073062-A None JP disclosed
JP-2073075-A None JP disclosed
EP-0006217-A1 Substituted amino acids, their use and preparation, and compositions containing them Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1980-01-09 EP disclosed
US-4139537-A 3-Aryloxy-1-(2- or 4-iminodihydro-1-pyridyl)-2-propanol antiarrhythmic compounds COOPER LABORATORIES, INC. (US) 1979-02-13 US disclosed