SCHEMBL6464047

SCHEMBL6464047

CC(c1cccc2ccccc12)[C@](N)(CC(=O)O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
EPHX2 P34913 2/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HIF1A Q16665 1/20 0.41
PTGER4 P35408 1/20 0.40
METAP2 P50579 1/20 0.40
METAP1 P53582 1/20 0.40
KIF11 P52732 1/20 0.39
SLC6A4 P31645 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALOX5 P09917 1/20 0.39
SSTR4 P31391 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1144334 0.76 CYP2C19 (0.58) CYP2C19HIF1AKIF11CYP1A2CYP2D6
SCHEMBL1144629 0.76 CYP2C19 (0.58) CYP2C19HIF1AKIF11CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL27488550 0.76 CYP2C9 (0.41) CYP2C9CYP2C19HPGDHDAC3HDAC1
SCHEMBL9848712 0.72 ALDH1A1 (0.47) CYP2C9CYP2C19HPGDHTTEPHX2
SCHEMBL27647539 0.71 ALOX5 (0.47) CYP2C9CYP2C19HDAC3HDAC1HDAC6
SCHEMBL9185404 0.70 CYP2C9 (0.59) CYP2C9CYP2C19HPGDHTTEPHX2
SCHEMBL2119043 0.70 PTGER4 (0.43) CYP2C9CYP2C19HPGDHTTEPHX2
SCHEMBL5328163 0.69 CYP2C9 (0.54) CYP2C9CYP2C19HPGDHTTEPHX2
SCHEMBL2242043 0.69 CYP1A2 (0.43) CYP2C9CYP2C19HPGDHTTHDAC3
SCHEMBL3814689 0.68 CYP2C9 (0.56) CYP2C9CYP2C19HPGDHTTEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493819-B1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER UBE INDUSTRIES (JP) 2014-11-12 EP disclosed
EP-1493819-A1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER Ube Industries, Ltd. (JP) 2005-01-05 EP disclosed