SCHEMBL6464059

SCHEMBL6464059

CC(c1cccc2ccccc12)C(c1ccccc1)[C@@H](N)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
SLC1A3 P43003 2/20 0.43
SLC1A2 P43004 2/20 0.43
SLC1A1 P43005 2/20 0.43
ALOX5 P09917 1/20 0.43
METAP2 P50579 3/20 0.41
METAP1 P53582 3/20 0.41
SLC6A4 P31645 1/20 0.40
ECE1 P42892 1/20 0.40
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
AKR1B1 P15121 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464051 1.00 ALDH1A1 (0.49) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL26966061 0.86 SLC1A3 (0.48) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL5326799 0.86 SLC1A3 (0.48) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL7366366 0.86 SLC1A3 (0.48) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL29628527 0.86 SLC1A3 (0.48) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL19682744 0.86 SLC1A3 (0.48) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL6460442 0.84 SLC1A3 (0.46) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL6460441 0.84 SLC1A3 (0.46) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL5283018 0.80 ALOX5 (0.46) ALDH1A1SLC1A3SLC1A2SLC1A1ALOX5
SCHEMBL5028930 0.77 ALOX5 (0.48) ALDH1A1ALOX5METAP2METAP1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1493819-B1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER UBE INDUSTRIES (JP) 2014-11-12 EP disclosed
EP-1493819-A1 PROCESS FOR PRODUCING EITHER OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID AND OPTICALLY ACTIVE N-SUBSTITUTED BETA-AMINO ACID ESTER OR OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID AND OPTICALLY ACTIVE N-SUBSTITUTED 2-HOMOPIPECOLIC ACID ESTER Ube Industries, Ltd. (JP) 2005-01-05 EP disclosed