Estradiol Methyl Ether

Estradiol Methyl Ether

SCHEMBL6464173

COc1ccc2c(c1)CC[C@@H]1[C@@H]2CC[C@@]2(C)[C@@H]1CC[C@@H]2O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 6/20 1.00
LMNA P02545 5/20 1.00
ESR1 P03372 6/20 0.77
SMN1; SMN2 Q16637 3/20 0.77
PGR P06401 2/20 0.77
AR P10275 2/20 0.77
SLC6A3 Q01959 2/20 0.77
ADORA3 P0DMS8 2/20 0.77
ATM Q13315 2/20 0.77
ABCC1 P33527 1/20 0.77
ABCC4 O15439 1/20 0.77
CHRM1 P11229 1/20 0.77
TBXA2R P21731 1/20 0.77
ADRA1A P35348 1/20 0.77
OPRM1 P35372 1/20 0.77
STS P08842 2/20 0.75
KDM4E B2RXH2 1/20 0.75
TSHR P16473 2/20 0.74
ESR2 Q92731 2/20 0.74
CYP2C9 P11712 2/20 0.74

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Estradiol Methyl Ether SCHEMBL12593628 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL14499084 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL8998255 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL15263441 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL547265 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL23645792 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL18686406 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL9558220 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
Estradiol Methyl Ether SCHEMBL4750578 1.00 HSD17B10 (1.00) HSD17B10LMNAESR1SMN1; SMN2PGR
SCHEMBL980768 0.92 LMNA (0.85) HSD17B10LMNAESR1SMN1; SMN2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6881728-B1 14-β, 17-α-hydroxymethylandrostane derivatives as androgens AKZO NOBEL N.V. (NL) 2005-04-19 US disclosed
EP-1163259-B1 14.BETA.,17-ALPHA-HYDROXYMETHYLANDROSTANE DERIVATIVES AS ANDROGENS AKZO NOBEL NV (NL) 2002-11-20 EP disclosed
EP-1163259-A1 14.BETA.,17-ALPHA-HYDROXYMETHYLANDROSTANE DERIVATIVES AS ANDROGENS Akzo Nobel N.V. (NL) 2001-12-19 EP disclosed
WO-2000053619-A1 14.BETA., 17-ALPHA-HYDROXYMETHYLANDROSTANE DERIVATIVES AS ANDROGENS AKZO NOBEL N.V. (NL) 2000-09-14 WO disclosed