SCHEMBL6464482

SCHEMBL6464482

CC(CNC(=O)O)CC(=O)NCCC(C(=O)c1nccs1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 3/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 2/20 0.35
CASR P41180 1/20 0.35
F11 P03951 1/20 0.35
RBBP9 O75884 1/20 0.34
HSPA9 P38646 2/20 0.34
HSPA5 P11021 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
MMP2 P08253 1/20 0.34
MMP3 P08254 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7043362 0.87 KCNA5 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6062401 0.82 L3MBTL1 (0.40) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6062993 0.82 EPHX2 (0.41) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6462336 0.82 HDAC1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6062741 0.80 EPHX2 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL7185649 0.77 ADORA2A (0.38) TSHREPHX2
SCHEMBL6676845 0.76 CYP1A2 (0.43) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL6467567 0.75 CTSS (0.38) CYP3A4CYP2D6CYP2C9CYP2C19LMNA
SCHEMBL7043168 0.69 MAPK1 (0.48) CYP3A4LMNAMAPK1SMN1; SMN2MMP2
SCHEMBL6475534 0.68 SMN1; SMN2 (0.39) CYP3A4CYP2D6CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed