SCHEMBL6465442

SCHEMBL6465442

COc1ccc(-c2nc(-c3ccc(O)c(OC)c3)[nH]c2-c2ccc(OC)cc2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOX1 Q9Y5S8 3/20 0.81
SMPD3 Q9NY59 4/20 0.79
MAPT P10636 7/20 0.63
TP53 P04637 4/20 0.63
MEN1 O00255 4/20 0.59
ALDH1A1 P00352 4/20 0.59
HPGD P15428 4/20 0.59
KMT2A Q03164 4/20 0.59
NPSR1 Q6W5P4 2/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
MAPK13 O15264 2/20 0.56
MAPK12 P53778 2/20 0.56
MAPK11 Q15759 2/20 0.56
MAPK14 Q16539 2/20 0.56
RAF1 P04049 1/20 0.56
KDM4E B2RXH2 3/20 0.56
CYP1A2 P05177 1/20 0.56
GLA P06280 1/20 0.56
GAA P10253 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6466286 0.89 NOX1 (0.72) NOX1SMPD3MAPTTP53MEN1
SCHEMBL6466417 0.88 NOX1 (0.79) NOX1SMPD3MAPTTP53MAPK13
SCHEMBL6691401 0.88 SMPD3 (1.00) NOX1SMPD3MAPTTP53MEN1
SCHEMBL6465425 0.88 SMPD3 (0.76) NOX1SMPD3MAPTTP53MEN1
SCHEMBL5676205 0.86 NOX1 (0.76) NOX1SMPD3MAPTTP53CYP1A2
SCHEMBL10588313 0.85 NOX1 (0.74) NOX1SMPD3MAPTTP53MEN1
SCHEMBL6469484 0.84 NOX1 (0.88) NOX1SMPD3MAPTTP53MAPK13
SCHEMBL6466475 0.83 NOX1 (0.71) NOX1SMPD3MAPTTP53MAPK13
SCHEMBL15400824 0.83 NOX1 (0.85) NOX1SMPD3MAPTTP53MEN1
SCHEMBL8008805 0.83 NOX1 (0.85) NOX1SMPD3MAPTTP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections AXXIMA PHARMACEUTICAL AG. (DE) 2005-09-15 US claimed
EP-1532118-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS Axxima Pharmaceuticals Aktiengesellschaft (DE) 2005-05-25 EP claimed
WO-2004005264-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS AXXIMA PHARMACEUTICALS AG (DE) 2004-01-15 WO claimed
US-20240000821-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER UNIV JOHNS HOPKINS (US) 2024-01-04 US disclosed
US-20200078387-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER THE JOHNS HOPKINS UNIVERSITY 2020-03-12 US disclosed
WO-2018112342-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2018-06-21 WO disclosed
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections AXXIMA PHARMACEUTICAL AG. (DE) 2005-09-15 US disclosed
EP-1532118-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS Axxima Pharmaceuticals Aktiengesellschaft (DE) 2005-05-25 EP disclosed
WO-2004005264-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS AXXIMA PHARMACEUTICALS AG (DE) 2004-01-15 WO disclosed
EP-0603953-B1 Use of 4' of 5'-hydroxy and 4'- or 5'-alkoxy-substituted electron transfer agents in compositions, elements, test kits and analytical methods JOHNSON & JOHNSON CLIN DIAG (US) 1999-02-17 EP disclosed
EP-0462644-B1 Biologically active reagents prepared from carboxy-containing polymer, analytical element and methods of use JOHNSON & JOHNSON CLIN DIAG (US) 1995-10-18 EP disclosed
WO-1990009594-A2 WASH COMPOSITION, TEST KIT AND THEIR USE TO DETERMINE A HERPES SIMPLEX VIRAL ANTIGEN EASTMAN KODAK COMPANY (US) 1990-08-23 WO disclosed
EP-0382519-A2 Extraction composition, test kit and their use to extract or determine herpes simplex viral antigen EASTMAN KODAK COMPANY (US) 1990-08-16 EP disclosed
EP-0370694-A2 Diagnostic kit and method using a solid phase capture means for detecting nucleic acids EASTMAN KODAK COMPANY (US) 1990-05-30 EP disclosed
EP-0363110-A2 High pH extraction composition and its use to determine a chlamydial, gonococcal or herpes antigen Johnson & Johnson Clinical Diagnostics, Inc. (US) 1990-04-11 EP disclosed
EP-0363109-A2 Determination of a chlamydial or gonococcal antigen using a positively-charged ionically binding support Johnson & Johnson Clinical Diagnostics, Inc. (US) 1990-04-11 EP disclosed
EP-0363090-A2 Diagnostic test kit and method for determination of chlamydial or gonococcal antigens using a microporous membrane Johnson & Johnson Clinical Diagnostics, Inc. (US) 1990-04-11 EP disclosed
EP-0363106-A2 Use of cationic surfactant to extract the chlamydial major outer membrane protein antigen Johnson & Johnson Clinical Diagnostics, Inc. (US) 1990-04-11 EP disclosed
EP-0363108-A2 Wash solution containing a cationic surfactant and its use in chlamydial and gonococcal determinations EASTMAN KODAK COMPANY (a New Jersey corporation) (US) 1990-04-11 EP disclosed
EP-0363089-A2 Use of a protease in the extraction of chlamydial, gonococcal and herpes antigens Johnson & Johnson Clinical Diagnostics, Inc. (US) 1990-04-11 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections CSNK1G1, CSNK1E, CSNK1D NOX1 2876/4885SMPD3 3746/4885MAPT 1480/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.