SCHEMBL6465479

SCHEMBL6465479

O=C(O)NCCCCC(=O)NCC(O)(CCc1ccccc1)c1nc(C(=O)NCc2ccccn2)co1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.46
ALOX15 P16050 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
SLC40A1 Q9NP59 4/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPK1 P28482 2/20 0.38
KMT2A Q03164 2/20 0.38
RAB9A P51151 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
KDM4E B2RXH2 2/20 0.38
POLB P06746 1/20 0.38
CYP2C9 P11712 1/20 0.38
MEN1 O00255 1/20 0.38
CYP2C19 P33261 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6465290 0.87 CYP3A4 (0.46) SMN1; SMN2ALDH1A1MAPK1KMT2ARAB9A
SCHEMBL7049145 0.78 KCNA5 (0.38) HPGDALOX15TDP1SLC40A1SMN1; SMN2
SCHEMBL6466215 0.73 SMN1; SMN2 (0.42) HPGDALOX15TDP1SLC40A1SMN1; SMN2
SCHEMBL4067173 0.66 HPGD (1.00) HPGDALOX15TDP1SMN1; SMN2ALDH1A1
SCHEMBL12125320 0.64 SMN1; SMN2 (0.80) HPGDALOX15TDP1SMN1; SMN2ALDH1A1
SCHEMBL18781735 0.64 SLC40A1 (0.62) HPGDSLC40A1SMN1; SMN2ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL29505709 0.63 SLC40A1 (0.62) HPGDSLC40A1SMN1; SMN2ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL18765428 0.63 SLC40A1 (0.62) HPGDSLC40A1SMN1; SMN2ALDH1A1MAPK1
SCHEMBL2840152 0.63 SMN1; SMN2 (0.56) HPGDALOX15TDP1SMN1; SMN2ALDH1A1
SCHEMBL1171725 0.63 EPHX2 (0.68) HPGDALOX15TDP1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed