SCHEMBL6467375

SCHEMBL6467375

COc1ccc(-c2nc(-c3cccc4ccccc34)[nH]c2-c2ccc(OC)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 3/20 0.62
MAPK12 P53778 3/20 0.62
MAPK11 Q15759 3/20 0.62
MAPK14 Q16539 3/20 0.62
GCGR P47871 2/20 0.62
MAPT P10636 4/20 0.60
TP53 P04637 2/20 0.60
RAF1 P04049 1/20 0.60
NOX1 Q9Y5S8 1/20 0.58
PDE10A Q9Y233 1/20 0.56
KDM4E B2RXH2 2/20 0.56
MEN1 O00255 2/20 0.56
ALDH1A1 P00352 2/20 0.56
HPGD P15428 2/20 0.56
KMT2A Q03164 2/20 0.56
CYP1A2 P05177 1/20 0.56
GLA P06280 1/20 0.56
GAA P10253 1/20 0.56
CYP2C19 P33261 1/20 0.56
GFER P55789 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17133338 0.89 MAPT (0.68) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL17133350 0.86 MAPT (0.73) MAPK13MAPK12MAPK11MAPK14MAPT
SCHEMBL2951436 0.84 MAPK14 (0.69) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL6465022 0.84 NOX1 (0.54) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL25272570 0.83 TEK (0.73) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL3194058 0.83 TEK (0.73) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL11082627 0.83 TEK (0.73) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL6466740 0.82 MAPK14 (0.67) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL5571856 0.82 NT5E (0.74) MAPK13MAPK12MAPK11MAPK14GCGR
SCHEMBL7989059 0.82 MAPT (0.51) MAPK13MAPK12MAPK11MAPK14GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections AXXIMA PHARMACEUTICAL AG. (DE) 2005-09-15 US claimed
EP-1532118-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS Axxima Pharmaceuticals Aktiengesellschaft (DE) 2005-05-25 EP claimed
WO-2004005264-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS AXXIMA PHARMACEUTICALS AG (DE) 2004-01-15 WO claimed
US-20240000821-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER UNIV JOHNS HOPKINS (US) 2024-01-04 US disclosed
US-20200078387-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER THE JOHNS HOPKINS UNIVERSITY 2020-03-12 US disclosed
WO-2018112342-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2018-06-21 WO disclosed
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections AXXIMA PHARMACEUTICAL AG. (DE) 2005-09-15 US disclosed
US-6903133-B2 Anticancer compounds PLANTACEUTICA, INC. (US) 2005-06-07 US disclosed
EP-1532118-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS Axxima Pharmaceuticals Aktiengesellschaft (DE) 2005-05-25 EP disclosed
US-20040138288-A1 Podophyllotoxin derivatives comprising furo[3',4':6,7]-naphtho[2,3-d]-1,3-dioxole ring; topoisomerase inhibitors PLANTACEUTICA, INC. 2004-07-15 US disclosed
WO-2004005264-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS AXXIMA PHARMACEUTICALS AG (DE) 2004-01-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections CSNK1G1, CSNK1E, CSNK1D MAPK13 456/4885MAPK12 732/4885MAPK11 1215/4885
US-20040138288-A1 Podophyllotoxin derivatives comprising furo[3',4':6,7]-naphtho[2,3-d]-1,3-dioxole ring; topoisomerase inhibitors TOP2A, TOP2B, TOP1 MAPK13 4581/4885MAPK12 4655/4885MAPK11 3924/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.