SCHEMBL64676

SCHEMBL64676

CCOC(=O)C1CN(C(=O)OCc2ccccc2)C(CO[Si](C)(C)C(C)(C)C)CC1OS(=O)(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
POLB P06746 1/20 0.35
ALDH1A1 P00352 2/20 0.35
PKM P14618 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65686 0.82 PDK1 (0.38) PDK1PDK2PDK3PDK4POLB
SCHEMBL9384838 0.79 ABCB1 (0.40) PDK1PDK2PDK3PDK4POLB
SCHEMBL65232 0.79 TMEM97 (0.37) PDK1PDK2PDK3PDK4POLB
SCHEMBL18740344 0.79 CYP2C19 (0.42) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL15341340 0.78 PDK1 (0.45) PDK1PDK2PDK3PDK4POLB
SCHEMBL8699830 0.78 POLB (0.49) PDK1PDK2PDK3PDK4POLB
SCHEMBL13340947 0.78 POLB (0.49) PDK1PDK2PDK3PDK4POLB
SCHEMBL1058641 0.78 POLB (0.49) PDK1PDK2PDK3PDK4POLB
SCHEMBL1058639 0.78 POLB (0.49) PDK1PDK2PDK3PDK4POLB
SCHEMBL5765731 0.77 ELANE (0.40) POLBMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed