SCHEMBL65686

SCHEMBL65686

CCOC(=O)C1CN(C(=O)OCc2ccccc2)C(CO[Si](C)(C)C(C)(C)C)CC1c1ccc(O)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
KDM1A O60341 1/20 0.37
RCOR1 Q9UKL0 1/20 0.37
HTR2C P28335 1/20 0.37
POLB P06746 1/20 0.36
PDE4B Q07343 1/20 0.35
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
CHRM2 P08172 2/20 0.35
CHRM4 P08173 2/20 0.35
CHRM5 P08912 2/20 0.35
CHRM1 P11229 2/20 0.35
CHRM3 P20309 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65232 0.89 TMEM97 (0.37) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL64234 0.86 L3MBTL1 (0.36) PDK1PDK2PDK3PDK4MAPT
SCHEMBL64057 0.86 PPARG (0.39) PDE4BMAPTCHRM2CHRM4CHRM5
SCHEMBL64676 0.82 PDK1 (0.39) PDK1PDK2PDK3PDK4POLB
SCHEMBL15341340 0.82 PDK1 (0.45) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL66855 0.81 ELANE (0.38) KDM1ARCOR1
SCHEMBL1058641 0.80 POLB (0.49) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL1058639 0.80 POLB (0.49) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL8699830 0.80 POLB (0.49) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL13340947 0.80 POLB (0.49) PDK1PDK2PDK3PDK4HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed