SCHEMBL6467665

SCHEMBL6467665

COCCN(CCOC)C(=O)N[C@@H](CS(=O)(=O)Cc1c(C)noc1C)C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.34
KMT2A Q03164 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
ALDH1A1 P00352 4/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
MEN1 O00255 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6467670 0.80 TDP1 (0.33) ARKMT2ATDP1SMN1; SMN2ALDH1A1
SCHEMBL7535471 0.74 CNR2 (0.36) KMT2ASMN1; SMN2ALDH1A1MEN1
SCHEMBL7415354 0.64 TDP1 (0.43) ARKMT2ATDP1ALDH1A1CYP1A2
SCHEMBL14378250 0.62 CYP1A2 (0.53) ARKMT2ATDP1ALDH1A1CYP1A2
SCHEMBL14426993 0.59 CYP1A2 (0.49) ARKMT2ATDP1ALDH1A1CYP1A2
SCHEMBL24811590 0.58 SMN1; SMN2 (0.41) KMT2ATDP1SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL1272532 0.58 CYP1A2 (0.54) ARKMT2ATDP1ALDH1A1CYP1A2
SCHEMBL18255993 0.57 P2RX7 (0.49) KMT2AALDH1A1MEN1L3MBTL1
SCHEMBL5013527 0.57 CYP1A2 (0.43) KMT2ATDP1ALDH1A1CYP1A2CYP3A4
SCHEMBL14759859 0.57 P2RX7 (0.48) KMT2ATDP1ALDH1A1MEN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed