SCHEMBL6468199

SCHEMBL6468199

COC(=O)c1cc(C(=O)O)cc(N(C)S(C)(=O)=O)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 4/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
TSHR P16473 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ALOX15 P16050 1/20 0.39
HIF1A Q16665 1/20 0.39
MAPK1 P28482 3/20 0.36
KDM6B O15054 1/20 0.35
KDM5C P41229 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM2A Q9Y2K7 1/20 0.35
KDM3A Q9Y4C1 1/20 0.35
BACE1 P56817 3/20 0.35
NQO2 P16083 1/20 0.34
USP2 O75604 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2711071 0.93 KMT2A (0.36) KMT2AKDM4EL3MBTL1TSHRALDH1A1
SCHEMBL2712407 0.84 KMT2A (0.37) KMT2AKDM4EL3MBTL1TSHRALDH1A1
SCHEMBL3510503 0.84 ALOX15 (0.44) KMT2AKDM4EL3MBTL1TSHRALDH1A1
SCHEMBL2711076 0.81 KMT2A (0.35) KMT2AKDM4EL3MBTL1TSHRALDH1A1
SCHEMBL21144538 0.78 TSHR (0.61) KDM4EL3MBTL1TSHRALDH1A1LMNA
SCHEMBL2021183 0.77 TTR (0.38) KMT2AKDM4ETSHRALDH1A1MEN1
SCHEMBL2018841 0.76 KDM4E (0.42) KMT2AKDM4EL3MBTL1TSHRALDH1A1
SCHEMBL11956572 0.75 TSHR (0.69) KDM4EL3MBTL1TSHRALDH1A1LMNA
SCHEMBL165562 0.74 KDM4E (0.51) KMT2AKDM4EL3MBTL1TSHRALDH1A1
SCHEMBL2719086 0.72 ALOX15 (0.48) KMT2AKDM4EL3MBTL1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed