SCHEMBL6468229

SCHEMBL6468229

Cc1csc(C2CCCN2C(=O)c2cc(-c3nnc(C(C)(Cc4ccccc4)NC(=O)OC(C)(C)C)o3)cc(N(C)S(C)(=O)=O)n2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.37
USP30 Q70CQ3 3/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.34
ACE P12821 1/20 0.32
TRPV1 Q8NER1 2/20 0.32
CPT2 P23786 1/20 0.32
CPT1A P50416 1/20 0.32
CPT1B Q92523 1/20 0.32
KLK5 Q9Y337 1/20 0.32
CPS1 P31327 1/20 0.31
POLB P06746 1/20 0.31
UCHL1 P09936 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
TRPC3 Q13507 1/20 0.30
TRPC6 Q9Y210 1/20 0.30
PKM P14618 1/20 0.30
MAPT P10636 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2725547 0.95 BACE1 (0.39) BACE1USP30BACE2SMN1; SMN2TRPV1
SCHEMBL2727474 0.89 BACE1 (0.48) BACE1USP30BACE2TRPV1CPT2
SCHEMBL2727473 0.89 BACE1 (0.48) BACE1USP30BACE2TRPV1CPT2
SCHEMBL6465415 0.89 BACE1 (0.48) BACE1USP30BACE2TRPV1CPT2
SCHEMBL6467781 0.88 SMN1; SMN2 (0.36) SMN1; SMN2ACETRPV1CPT2CPT1A
SCHEMBL6466800 0.87 SMN1; SMN2 (0.34) BACE1SMN1; SMN2ACETRPV1CPT2
SCHEMBL6468770 0.86 SMN1; SMN2 (0.37) SMN1; SMN2ACETRPV1CPT2CPT1A
SCHEMBL10289972 0.85 USP30 (0.37) USP30SMN1; SMN2ACETRPV1CPT2
SCHEMBL2725028 0.84 BACE1 (0.37) BACE1USP30BACE2SMN1; SMN2TRPV1
SCHEMBL2729431 0.83 CPT1A (0.40) SMN1; SMN2ACETRPV1CPT2CPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed