SCHEMBL6469273

SCHEMBL6469273

N#Cc1ccc(S(=O)(=O)CCN2CCCCC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.52
LOX P28300 4/20 0.50
HRH2 P25021 1/20 0.47
HRH1 P35367 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GAA P10253 2/20 0.46
MAPT P10636 1/20 0.46
KCNH2 Q12809 3/20 0.45
KCNJ1 P48048 1/20 0.45
TSHR P16473 1/20 0.43
SCN7A Q01118 1/20 0.43
LTA4H P09960 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6011962 0.82 HRH3 (0.51) HRH3LOXHRH2HRH1MEN1
SCHEMBL56319 0.80 LOX (0.57) HRH3LOXMEN1KMT2AGAA
SCHEMBL2921597 0.80 ESR1 (0.58) HRH3LOXMEN1KMT2AGAA
SCHEMBL13604236 0.79 KMT2A (0.71) LOXMEN1KMT2ALTA4H
SCHEMBL2922255 0.78 ESR1 (0.56) LOXMEN1KMT2AGAALTA4H
SCHEMBL14476103 0.77 MEN1 (0.73) LOXMEN1KMT2ALTA4H
SCHEMBL6837022 0.76 ALDH1A1 (0.51) HRH3LOXMEN1KMT2AKCNH2
SCHEMBL8412814 0.76 ESR1 (0.52) LOXMEN1KMT2AGAATSHR
SCHEMBL8423201 0.76 SMN1; SMN2 (0.60) HRH3LOXKMT2AGAAMAPT
SCHEMBL12015819 0.74 LOX (0.51) LOXMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1572650-A1 NOVEL PIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR CCR5 AstraZeneca AB (SE) 2005-09-14 EP disclosed
WO-2004056773-A1 NOVEL PIPERIDINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR CCR5 ASTRAZENECA AB (SE) 2004-07-08 WO disclosed