SCHEMBL6469885

SCHEMBL6469885

Oc1ccc(-c2nc(-c3ccncc3)c(-c3ccc(Cl)cc3)[nH]2)cc1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.86
MAPK13 O15264 14/20 0.86
MAPK12 P53778 14/20 0.86
MAPK11 Q15759 14/20 0.86
GCGR P47871 11/20 0.86
RAF1 P04049 7/20 0.77
BRAF P15056 3/20 0.77
CSNK1D P48730 3/20 0.75
MAPK9 P45984 3/20 0.75
CSNK1E P49674 2/20 0.75
PRKD3 O94806 2/20 0.75
MAP4K4 O95819 2/20 0.75
FRK P42685 2/20 0.75
CSNK1A1 P48729 2/20 0.75
GSK3B P49841 2/20 0.75
PTK6 Q13882 2/20 0.75
CLK4 Q9HAZ1 2/20 0.75
KDM4E B2RXH2 1/20 0.75
CIT O14578 1/20 0.75
GAK O14976 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6471005 0.93 MAPK13 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL29587593 0.93 CYP19A1 (0.72) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL2649730 0.93 MAPK13 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL5921859 0.87 MAPK13 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL6469111 0.87 MAPK13 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL28486758 0.87 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL6469877 0.87 MAPK14 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL8234546 0.86 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL2649616 0.86 MAPK13 (1.00) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL21557235 0.86 MAPK14 (0.77) MAPK14MAPK13MAPK12MAPK11GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections AXXIMA PHARMACEUTICAL AG. (DE) 2005-09-15 US claimed
US-20240000821-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER UNIV JOHNS HOPKINS (US) 2024-01-04 US disclosed
US-20200078387-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER THE JOHNS HOPKINS UNIVERSITY 2020-03-12 US disclosed
WO-2018112342-A1 CHEMICAL INHIBITORS AGAINST KINASES TO BLOCK TELOMERE ELONGATION IN CANCER THE JOHNS HOPKINS UNIVERSITY (US) 2018-06-21 WO disclosed
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections AXXIMA PHARMACEUTICAL AG. (DE) 2005-09-15 US disclosed
EP-1532118-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS Axxima Pharmaceuticals Aktiengesellschaft (DE) 2005-05-25 EP disclosed
WO-2004005264-A2 IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF HEPATITIS C VIRUS INFECTIONS AXXIMA PHARMACEUTICALS AG (DE) 2004-01-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050203155-A1 Imidazole compounds and human cellular proteins casein kinase I alpha, delta and epsilon as targets for medical intervention against Hepatitis C Virus infections CSNK1G1, CSNK1E, CSNK1D MAPK14 662/4885MAPK13 456/4885MAPK12 732/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.