SCHEMBL6470455

SCHEMBL6470455

NC(=O)C(O)=Cc1cccc(-c2ncc[nH]2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.47
MTOR P42345 1/20 0.47
ADK P55263 1/20 0.47
VCP P55072 4/20 0.45
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
PARP1 P09874 1/20 0.42
JAK3 P52333 2/20 0.42
RPS6KA5 O75582 1/20 0.42
CSNK1A1 P48729 1/20 0.42
TYRO3 Q06418 1/20 0.42
DYRK1B Q9Y463 1/20 0.42
MAP2K4 P45985 1/20 0.42
RPS6KA3 P51812 1/20 0.42
MELK Q14680 1/20 0.42
NEK2 P51955 2/20 0.39
ERBB2 P04626 1/20 0.38
TEC P42680 1/20 0.38
TXK P42681 1/20 0.38
BLK P51451 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6470451 1.00 NISCH (0.47) NISCHMTORADKVCPKDM4E
SCHEMBL29957239 0.77 NISCH (0.55) NISCHMTORADKVCPKDM4E
SCHEMBL4623510 0.77 NISCH (0.55) NISCHMTORADKVCPKDM4E
SCHEMBL5481767 0.76 PRKCI (0.55) NISCHMTORADKVCPKDM4E
SCHEMBL45099 0.74 KDM4E (0.68) NISCHMTORADKVCPKDM4E
SCHEMBL29569789 0.74 KDM4E (0.68) NISCHMTORADKVCPKDM4E
Oxalic Acid SCHEMBL31679099 0.73 MTOR (0.54) NISCHMTORADKVCPKDM4E
SCHEMBL6470431 0.73 HDAC1 (0.62) VCP
SCHEMBL6470430 0.73 HDAC1 (0.62) VCP
SCHEMBL16777437 0.73 NISCH (0.72) NISCHMTORADKVCPKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005065681-A1 N- HYDROXY-3-(3-(1H-IMIDAZOL-2-YL)-PHENYL)-ACRYLAMIDE DERIVATIVES AND RELATED COMPOUNDS AS HISTONE DEACETYLASE (HDAC) INHIBITORS FOR THE TREATMENT OF CANCER TAKEDA SAN DIEGO, INC. (US) 2005-07-21 WO disclosed