SCHEMBL6470827

SCHEMBL6470827

Nc1ccc(C=CC=O)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 1/20 0.45
TRPA1 O75762 2/20 0.43
LMNA P02545 1/20 0.43
ALOX5 P09917 1/20 0.43
MAPK1 P28482 1/20 0.43
XDH P47989 2/20 0.41
GABRP O00591 2/20 0.39
GABRD O14764 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRB1 P18505 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRA3 P34903 2/20 0.39
GABRA2 P47869 2/20 0.39
GABRB2 P47870 2/20 0.39
GABRA4 P48169 2/20 0.39
GABRE P78334 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16379657 1.00 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL25490677 0.80 NOS3 (0.39) ALDH1A1KDM4EGABRPGABRDGABRA1
SCHEMBL1637193 0.79
SCHEMBL29854831 0.79
SCHEMBL7899522 0.77 NOS3 (0.43) ALDH1A1KDM4EGABRPGABRDGABRA1
SCHEMBL18255135 0.76 KDM4E (0.45) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL6852107 0.76 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL6273189 0.76 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL18921523 0.76 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTTRPA1LMNA
SCHEMBL18921524 0.76 ALDH1A1 (0.45) ALDH1A1KDM4EMAPTTRPA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050107381-A1 6-membered heteroaryl compounds for the treatment of neurodegenerative disorders PFIZER, INC. 2005-05-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050107381-A1 6-membered heteroaryl compounds for the treatment of neurodegenerative disorders APP, BACE1, SNCA ALDH1A1 2820/4885KDM4E 3151/4885MAPT 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.