SCHEMBL6473192

SCHEMBL6473192

CCCCCOc1cc2c(cc1-c1cc(C=CC(=O)OCC)ccc1OCOC)C(C)(C)CCC2(C)C

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FDPS P14324 1/20 0.49
ACHE P22303 4/20 0.47
RXRA P19793 2/20 0.47
BCHE P06276 3/20 0.47
APP P05067 5/20 0.43
MAOB P27338 1/20 0.41
HPGD P15428 2/20 0.41
ALDH1A1 P00352 1/20 0.41
THRB P10828 1/20 0.41
CNR2 P34972 1/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TTR P02766 1/20 0.40
DPP4 P27487 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6473188 1.00 FDPS (0.49) FDPSACHERXRABCHEAPP
SCHEMBL6477392 0.95 FDPS (0.51) FDPSACHERXRABCHEAPP
SCHEMBL6477393 0.95 FDPS (0.51) FDPSACHERXRABCHEAPP
SCHEMBL6473193 0.90 RXRA (0.51) ACHERXRACNR2MEN1KMT2A
SCHEMBL6473191 0.90 RXRA (0.51) ACHERXRACNR2MEN1KMT2A
SCHEMBL6476811 0.90 FDPS (0.53) FDPSACHERXRABCHEMAOB
SCHEMBL6476815 0.90 FDPS (0.53) FDPSACHERXRABCHEMAOB
SCHEMBL6472649 0.87 RXRA (0.54) FDPSACHERXRABCHEAPP
SCHEMBL6472653 0.87 RXRA (0.54) FDPSACHERXRABCHEAPP
SCHEMBL6472405 0.87 KDM4E (0.47) FDPSRXRAAPPHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924388-B2 Bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-02 US disclosed
US-20040092594-A1 Bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-05-13 US disclosed
US-6632963-B1 Are useful for the treatment of a wide variety of disease states, whether human or veterinary, for example dermatological, rheumatic, respiratory, cardiovascular and ophthalmological disorders, as well as for the treatment of GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2003-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092594-A1 Bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof AHR, TYR, MC1R FDPS 3696/4885ACHE 2858/4885RXRA 174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.