SCHEMBL6473338

SCHEMBL6473338

Cn1c(=O)n(Cc2ccccc2)c(=O)c2c(C(=O)OCc3ccc([N+](=O)[O-])cc3)csc21

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
LMNA P02545 1/20 0.43
KMT2A Q03164 6/20 0.43
ALDH1A1 P00352 2/20 0.43
ATM Q13315 1/20 0.42
MEN1 O00255 4/20 0.42
POLB P06746 2/20 0.42
AR P10275 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
PLCG1 P19174 1/20 0.40
MAPT P10636 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6471284 0.91 MEN1 (0.46) RAB9ATDP1LMNAKMT2AALDH1A1
SCHEMBL6258578 0.88 ALDH1A1 (0.44) KMT2AALDH1A1MEN1POLBL3MBTL1
SCHEMBL6470730 0.87 TP53 (0.48) TDP1LMNAKMT2AALDH1A1MEN1
SCHEMBL6258893 0.86 MEN1 (0.42) RAB9AKMT2AMEN1POLBL3MBTL1
SCHEMBL6476368 0.86 MEN1 (0.44) KMT2AALDH1A1MEN1POLB
SCHEMBL6473171 0.85 MEN1 (0.41) RAB9ALMNAKMT2AALDH1A1MEN1
SCHEMBL7105782 0.85 MEN1 (0.41) RAB9ALMNAKMT2AALDH1A1MEN1
SCHEMBL6472338 0.85 MEN1 (0.41) LMNAKMT2AALDH1A1MEN1POLB
SCHEMBL6260852 0.84 NPSR1 (0.43) RAB9ALMNAKMT2AALDH1A1MEN1
SCHEMBL6470949 0.82 POLB (0.42) RAB9ALMNAKMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530475-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 AND A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006931-A2 PHARMACEUTICAL COMPOSTIONS COMPRISING AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 AND A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed