SCHEMBL6260852

SCHEMBL6260852

Cn1c(=O)n(Cc2ccccc2)c(=O)c2c(C(=O)OCc3ccc(Cl)c(Cl)c3)csc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
MEN1 O00255 6/20 0.42
KMT2A Q03164 6/20 0.42
MAPT P10636 5/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.41
ERCC5 P28715 1/20 0.39
FEN1 P39748 1/20 0.39
HIF1A Q16665 2/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MMP13 P45452 1/20 0.38
CYP3A4 P08684 2/20 0.38
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6471284 0.90 MEN1 (0.46) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL6258578 0.90 ALDH1A1 (0.44) NPSR1MEN1KMT2AMAPTPOLB
SCHEMBL6470998 0.88 POLB (0.42) MEN1KMT2AMAPTSMN1; SMN2POLB
SCHEMBL6473171 0.87 MEN1 (0.41) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL6470730 0.87 TP53 (0.48) NPSR1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL6472301 0.86 MMP1 (0.47) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL6257046 0.86 THRB (0.47) MEN1KMT2AMAPTSMN1; SMN2LMNA
SCHEMBL6476368 0.86 MEN1 (0.44) MEN1KMT2ASMN1; SMN2GAAPOLB
SCHEMBL6258893 0.86 MEN1 (0.42) MEN1KMT2ASMN1; SMN2GAAPOLB
SCHEMBL6253632 0.85 MEN1 (0.43) MEN1KMT2AMAPTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530467-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006912-A2 COMBINATION OF AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed