SCHEMBL6474567

SCHEMBL6474567

O=C(OCc1cnn[nH]1)c1ccncn1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.41
GRM4 Q14833 1/20 0.35
POLB P06746 2/20 0.34
CTNNB1 P35222 1/20 0.34
WNT3A P56704 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
SIRT3 Q9NTG7 1/20 0.34
KMT2A Q03164 1/20 0.33
MAPT P10636 1/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TSHR P16473 1/20 0.33
PKM P14618 1/20 0.33
TBXA2R P21731 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236586 0.73 TDP1 (0.54) P2RX7POLBKMT2ANPSR1TSHR
SCHEMBL7103527 0.72 P2RX7 (0.43) P2RX7GRM4CTNNB1WNT3AGAA
SCHEMBL917137 0.71 CYP1A2 (0.53) P2RX7CTNNB1WNT3AKMT2AMAPT
SCHEMBL29508230 0.71 CYP1A2 (0.53) P2RX7CTNNB1WNT3AKMT2AMAPT
SCHEMBL31722590 0.71 P2RX7 (0.51) P2RX7GRM4CTNNB1WNT3AKMT2A
SCHEMBL27846622 0.71 P2RX7 (0.51) P2RX7GRM4POLBCTNNB1WNT3A
SCHEMBL27798556 0.71 P2RX7 (0.56) P2RX7GRM4CTNNB1WNT3ASIRT2
SCHEMBL27902698 0.71 SNCA (0.52) P2RX7GRM4CTNNB1WNT3AKMT2A
SCHEMBL7017659 0.70 P2RX7 (0.41) P2RX7GRM4POLBCTNNB1WNT3A
Hydrochloric Acid SCHEMBL27922723 0.70 CYP1A2 (0.51) P2RX7CTNNB1WNT3AKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530475-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 AND A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006931-A2 PHARMACEUTICAL COMPOSTIONS COMPRISING AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 AND A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed