SCHEMBL7103527

SCHEMBL7103527

O=C(OCc1ncc[nH]1)c1ccncn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.43
TBXAS1 P24557 2/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 2/20 0.36
HTT P42858 1/20 0.36
CTNNB1 P35222 1/20 0.35
WNT3A P56704 1/20 0.35
CYP3A4 P08684 1/20 0.34
TAAR1 Q96RJ0 2/20 0.34
FDPS P14324 1/20 0.34
GRM4 Q14833 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
FPR2 P25090 1/20 0.34
PKM P14618 1/20 0.34
TBXA2R P21731 2/20 0.33
HTR1A P08908 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236586 0.75 TDP1 (0.54) P2RX7CYP3A4NPSR1PKMALDH1A1
SCHEMBL29508230 0.73 CYP1A2 (0.53) P2RX7KDM4ECTNNB1WNT3AALDH1A1
SCHEMBL27846622 0.73 P2RX7 (0.51) P2RX7KDM4EGAACTNNB1WNT3A
SCHEMBL917137 0.73 CYP1A2 (0.53) P2RX7KDM4ECTNNB1WNT3AALDH1A1
SCHEMBL27798556 0.73 P2RX7 (0.56) P2RX7CTNNB1WNT3AGRM4NPSR1
SCHEMBL31722590 0.73 P2RX7 (0.51) P2RX7KDM4EGAACTNNB1WNT3A
SCHEMBL6474567 0.72 P2RX7 (0.41) P2RX7GAACTNNB1WNT3AGRM4
Hydrochloric Acid SCHEMBL27922723 0.72 CYP1A2 (0.51) P2RX7KDM4ECTNNB1WNT3AALDH1A1
SCHEMBL21624605 0.72 TBXAS1 (0.44) TBXAS1GAACYP3A4TAAR1FDPS
SCHEMBL6432861 0.72 FDPS (0.45) TBXAS1KDM4EGAAHTTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370562-A1 THIENO[2,3-D]PYRIMIDINDIONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2003-12-17 EP claimed
WO-2002064598-A1 THIENO'2,3-D PYRIMIDINDIONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2002-08-22 WO claimed