SCHEMBL6474779

SCHEMBL6474779

COc1ccc(-c2ccccc2)c2sc(NC(=O)c3ccc(CNC4CCCC4)cc3)nc12

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.49
CHRM4 P08173 2/20 0.48
DUSP3 P51452 2/20 0.48
MAPT P10636 3/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ADORA2A P29274 9/20 0.45
ADORA2B P29275 9/20 0.45
ADORA1 P30542 9/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3037638 0.99 HDAC1 (0.48) HDAC1CHRM4DUSP3MAPTALDH1A1
SCHEMBL6482561 0.98 DUSP3 (0.48) HDAC1CHRM4DUSP3MAPTALDH1A1
Hydrochloric Acid SCHEMBL3047354 0.97 DUSP3 (0.47) HDAC1CHRM4DUSP3MAPTALDH1A1
SCHEMBL6476610 0.87 DUSP3 (0.48) HDAC1CHRM4DUSP3MAPTALDH1A1
SCHEMBL6476277 0.86 DUSP3 (0.53) CHRM4DUSP3ADORA2AADORA2BADORA1
Hydrochloric Acid SCHEMBL3057668 0.86 DUSP3 (0.48) HDAC1CHRM4DUSP3MAPTALDH1A1
Hydrochloric Acid SCHEMBL3045899 0.86 DUSP3 (0.53) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL3046423 0.85 DUSP3 (0.56) CHRM4DUSP3ADORA2AADORA2BADORA1
SCHEMBL6477408 0.85 DUSP3 (0.52) CHRM4DUSP3ALDH1A1ADORA2AADORA2B
SCHEMBL6476606 0.84 ADORA2B (0.50) CHRM4DUSP3MAPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed