SCHEMBL6475799

SCHEMBL6475799

COc1ccc(-c2ccccc2)c2sc(NC(=O)c3ccc(CN4CCOCC4)cc3)nc12

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.57
MEN1 O00255 2/20 0.57
MAPT P10636 4/20 0.56
ADORA2A P29274 3/20 0.53
ADORA1 P30542 3/20 0.53
ADORA2B P29275 2/20 0.53
HIF1A Q16665 2/20 0.52
EPAS1 Q99814 2/20 0.52
HDAC1 Q13547 2/20 0.52
HDAC6 Q9UBN7 1/20 0.52
SMN1; SMN2 Q16637 2/20 0.50
MAPK1 P28482 2/20 0.50
NPC1 O15118 1/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
RAB9A P51151 1/20 0.50
GAA P10253 1/20 0.50
ALK Q9UM73 1/20 0.48
TRPV4 Q9HBA0 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3046550 0.99 KMT2A (0.56) KMT2AMEN1MAPTADORA2AADORA1
SCHEMBL5036546 0.92 HDAC1 (0.54) KMT2AMEN1MAPTADORA2AADORA1
Hydrochloric Acid SCHEMBL3048068 0.91 HDAC1 (0.54) KMT2AMEN1MAPTADORA2AADORA1
SCHEMBL6485716 0.91 HDAC1 (0.54) KMT2AMEN1MAPTADORA2AADORA1
SCHEMBL3039082 0.91 HDAC1 (0.53) KMT2AMEN1MAPTADORA2AADORA1
SCHEMBL6481675 0.91 ALK (0.54) MAPTADORA2AADORA1ADORA2BHDAC1
Hydrochloric Acid SCHEMBL3051261 0.91 TRPV4 (0.53) KMT2AMEN1MAPTADORA2AADORA1
SCHEMBL6476780 0.90 HDAC1 (0.52) KMT2AMEN1MAPTADORA2AADORA1
Hydrochloric Acid SCHEMBL3048499 0.90 HDAC1 (0.52) KMT2AMEN1MAPTADORA2AADORA1
Hydrochloric Acid SCHEMBL3053390 0.90 KIT (0.53) MAPTADORA2AADORA1ADORA2BHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed