SCHEMBL6476291

SCHEMBL6476291

COc1ccc(-c2ccccc2)c2sc(NC(=O)c3ccc(CN(C)Cc4cccnc4)cc3)nc12

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 3/20 0.54
TP53 P04637 4/20 0.49
MAPT P10636 3/20 0.49
ADORA2A P29274 6/20 0.48
ADORA2B P29275 6/20 0.48
ADORA1 P30542 6/20 0.48
DUSP3 P51452 1/20 0.46
HIF1A Q16665 1/20 0.45
EPAS1 Q99814 1/20 0.45
LMNA P02545 1/20 0.45
POLB P06746 1/20 0.45
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3037965 0.99 CHRM4 (0.53) CHRM4TP53MAPTADORA2AADORA2B
SCHEMBL6481259 0.93 ADORA2B (0.53) CHRM4ADORA2AADORA2BADORA1DUSP3
Hydrochloric Acid SCHEMBL3048033 0.92 ADORA2B (0.53) CHRM4ADORA2AADORA2BADORA1DUSP3
SCHEMBL3049501 0.88 CHRM4 (0.55) CHRM4TP53MAPTADORA2AADORA2B
Hydrochloric Acid SCHEMBL3042509 0.88 CHRM4 (0.54) CHRM4TP53MAPTADORA2AADORA2B
SCHEMBL6486465 0.87 ADORA2B (0.54) CHRM4ADORA2AADORA2BADORA1DUSP3
SCHEMBL6483836 0.86 ADORA2B (0.53) CHRM4ADORA2AADORA2BADORA1DUSP3
Hydrochloric Acid SCHEMBL3059825 0.86 ADORA2B (0.53) CHRM4ADORA2AADORA2BADORA1DUSP3
Hydrochloric Acid SCHEMBL3043464 0.86 ADORA2B (0.52) CHRM4ADORA2AADORA2BADORA1DUSP3
SCHEMBL3049496 0.85 TP53 (0.52) CHRM4TP53MAPTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed