SCHEMBL6478035

SCHEMBL6478035

C#Cc1ccc(OCOC)c(-c2cc3c(cc2C)C(C)(C)CCC3(C)C)c1

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RARG P13631 13/20 0.42
RARB P10826 4/20 0.38
RARA P10276 3/20 0.38
RXRA P19793 7/20 0.36
RXRG P48443 3/20 0.36
RXRB P28702 2/20 0.36
PPARG P37231 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6473292 0.83 RARG (0.47) RARGRARBRARARXRARXRG
SCHEMBL6473301 0.81 RARG (0.42) RARGRARBRARARXRARXRG
SCHEMBL6880773 0.75 RARG (0.49) RARGRARBRARARXRARXRG
SCHEMBL6880775 0.74 RXRA (0.67) RARGRXRARXRGRXRB
SCHEMBL6869561 0.71 RARG (0.46) RARGRARBRARARXRARXRG
SCHEMBL1629484 0.71 AR (0.36)
SCHEMBL6472962 0.71 RXRA (0.56) RARGRARBRARARXRARXRG
SCHEMBL6472965 0.71 RXRA (0.56) RARGRARBRARARXRARXRG
SCHEMBL6875617 0.70 RXRA (0.45) RARGRARBRARARXRARXRG
SCHEMBL6876532 0.68 RARG (0.49) RARGRARBRARARXRARXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924388-B2 Bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-02 US disclosed
US-20040092594-A1 Bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-05-13 US disclosed
US-6632963-B1 Are useful for the treatment of a wide variety of disease states, whether human or veterinary, for example dermatological, rheumatic, respiratory, cardiovascular and ophthalmological disorders, as well as for the treatment of GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2003-10-14 US disclosed
EP-0947496-A1 Bicyclic aromatic compounds and their use in human and veterinary medicine as well as in cosmetology Galderma Research & Development, S.N.C. (FR) 1999-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092594-A1 Bicyclic aromatic compounds and pharmaceutical/cosmetic compositions comprised thereof AHR, TYR, MC1R RARG 302/4885RARB 328/4885RARA 198/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.