SCHEMBL6479159

SCHEMBL6479159

Cc1c[nH]nc1S(=O)(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccc(OC(=O)N(C)C)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 6/20 0.44
ITGB1 P05556 12/20 0.43
ITGA4 P13612 8/20 0.43
ITGB7 P26010 1/20 0.43
ITGAV P06756 3/20 0.38
ITGA5 P08648 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3852356 0.91 CACNA1B (0.45) CACNA1BITGB1ITGA4ITGB7ITGAV
SCHEMBL5608873 0.86 ITGB1 (0.44) CACNA1BITGB1ITGA4ITGB7ITGAV
SCHEMBL3855808 0.86 ITGA4 (0.52) CACNA1BITGB1ITGA4ITGB7ITGA5
SCHEMBL3851264 0.85 CACNA1B (0.51) CACNA1BITGB1ITGA4ITGB7ITGA5
SCHEMBL3855039 0.84 CACNA1B (0.46) CACNA1BITGB1ITGA4ITGB7ITGA5
SCHEMBL3855409 0.84 ITGB1 (0.46) CACNA1BITGB1ITGA4ITGB7ITGAV
SCHEMBL4451846 0.83 KDM4E (0.43) CACNA1BITGB1ITGA4ITGB7
SCHEMBL3855049 0.83 CACNA1B (0.46) CACNA1BITGB1ITGA4ITGB7ITGAV
SCHEMBL12317079 0.83 ITGB1 (0.48) CACNA1BITGB1ITGA4ITGB7ITGAV
SCHEMBL3855802 0.83 CACNA1B (0.46) CACNA1BITGB1ITGA4ITGB7ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900179-B2 Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. 2005-05-31 US disclosed
US-20020193312-A1 Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. 2002-12-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020193312-A1 Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4 VCAM1, ICAM1, L1CAM CACNA1B 383/4885ITGB1 64/4885ITGA4 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.