SCHEMBL6479950

SCHEMBL6479950

CC1S[C@H]2C[C@@](Cc3ccccc3)(NC(=O)OC(C)(C)C)C(=O)N2[C@@H]1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPIA P62937 1/20 0.39
GRIN2B Q13224 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SCN9A Q15858 3/20 0.35
AKT1 P31749 4/20 0.34
ATM Q13315 1/20 0.34
CTSK P43235 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
DPP9 Q86TI2 1/20 0.34
CTSL P07711 1/20 0.33
ACE P12821 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6474085 0.83 GFER (0.32)
SCHEMBL6479934 0.83 GFER (0.32)
SCHEMBL1728442 0.82 PPIA (0.39) PPIAGRIN2BCA12CA1CA7
SCHEMBL1730102 0.79 DPP4 (0.40) PPIAGRIN2BCA12CA1CA7
SCHEMBL6479943 0.79 PPIA (0.40) PPIAGRIN2BCA12CA1CA7
SCHEMBL1728443 0.79 PPIA (0.40) PPIAGRIN2BCA12CA1CA7
SCHEMBL1730373 0.77 PPIA (0.41) PPIAGRIN2BCA12CA1CA7
SCHEMBL7411070 0.72 BRD4 (0.40) PPIAGRIN2BCA12CA1CA7
SCHEMBL8225058 0.70 F2 (0.47) PPIACA12CA1CA7CA14
SCHEMBL8227078 0.70 F2 (0.47) PPIACA12CA1CA7CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050059716-A1 Novel bicyclic cyanoheterocycles, process for their preparation and their use as medicaments AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2005-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059716-A1 Novel bicyclic cyanoheterocycles, process for their preparation and their use as medicaments CYP11B2, GOT2, CYP11B1 PPIA 934/4885GRIN2B 761/4885CA12 724/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.