SCHEMBL6482952

SCHEMBL6482952

CCN(CC)Cc1ccc(C(=O)Nc2nc3c(OC)ccc(-c4ccccc4)c3s2)cc1

nearest known ligand 0.55

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.55
ADORA2B P29275 16/20 0.55
ADORA1 P30542 16/20 0.55
DUSP3 P51452 1/20 0.51
CHRM4 P08173 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3044718 0.99 ADORA2A (0.54) ADORA2AADORA2BADORA1DUSP3CHRM4
SCHEMBL6476220 0.93 ADORA2A (0.51) ADORA2AADORA2BADORA1DUSP3CHRM4
Hydrochloric Acid SCHEMBL3048459 0.92 ADORA2A (0.51) ADORA2AADORA2BADORA1DUSP3CHRM4
SCHEMBL6486465 0.91 ADORA2B (0.54) ADORA2AADORA2BADORA1DUSP3CHRM4
Hydrochloric Acid SCHEMBL3059825 0.90 ADORA2B (0.53) ADORA2AADORA2BADORA1DUSP3CHRM4
SCHEMBL6481259 0.90 ADORA2B (0.53) ADORA2AADORA2BADORA1DUSP3CHRM4
Hydrochloric Acid SCHEMBL3048033 0.89 ADORA2B (0.53) ADORA2AADORA2BADORA1DUSP3CHRM4
SCHEMBL3053634 0.89 DUSP3 (0.54) ADORA2AADORA2BADORA1DUSP3CHRM4
SCHEMBL3046423 0.88 DUSP3 (0.56) ADORA2AADORA2BADORA1DUSP3CHRM4
SCHEMBL7198817 0.88 ADORA2A (0.51) ADORA2AADORA2BADORA1DUSP3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6963000-B2 Benzothiazole derivatives with activity as adenosine receptor ligands HOFFMAN-LA ROCHE INC. (US) 2005-11-08 US claimed