SCHEMBL6487292

SCHEMBL6487292

COC(=O)[C@H]1CNCCN1C(=O)OCc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.52
PREP P48147 3/20 0.49
NPSR1 Q6W5P4 1/20 0.49
FKBP1A P62942 1/20 0.47
ALDH1A1 P00352 1/20 0.47
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TP53 P04637 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TSHR P16473 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
CTSK P43235 1/20 0.46
GFER P55789 1/20 0.45
CTRB1 P17538 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3017853 1.00 HTR2C (0.52) HTR2CPREPNPSR1FKBP1AALDH1A1
SCHEMBL6501753 1.00 HTR2C (0.52) HTR2CPREPNPSR1FKBP1AALDH1A1
Hydrochloric Acid SCHEMBL7013165 0.99 HTR2C (0.51) HTR2CPREPNPSR1FKBP1AALDH1A1
Trifluoroacetic Acid SCHEMBL30253251 0.94 HTR2C (0.46) HTR2CPREPNPSR1FKBP1AALDH1A1
SCHEMBL4674934 0.91 HTR2C (0.52) HTR2CPREPNPSR1FKBP1ANPC1
SCHEMBL27736628 0.89 HTR2C (0.51) HTR2CPREPNPSR1FKBP1ATSHR
SCHEMBL27757498 0.89 HTR2C (0.51) HTR2CPREPNPSR1FKBP1ATSHR
SCHEMBL20299652 0.89 FKBP1A (0.52) HTR2CPREPNPSR1FKBP1AALDH1A1
SCHEMBL7251746 0.88 HTR2C (0.53) HTR2CPREPNPSR1NPC1RAB9A
SCHEMBL8220722 0.88 HTR2C (0.53) HTR2CPREPNPSR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6911442-B1 Quinoline derivatives as antibacterials SMITHKLINE BEECHAM P.L.C. (GB) 2005-06-28 US disclosed
EP-1187828-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2004-04-21 EP disclosed
EP-1187828-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2002-03-20 EP disclosed
WO-2000078748-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-28 WO disclosed