SCHEMBL6489735

SCHEMBL6489735

O=C1CC(C(=O)N2CCC(c3ccccc3)CC2)Cc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.48
HTR2B P41595 1/20 0.46
NAMPT P43490 5/20 0.46
CYP19A1 P11511 1/20 0.45
GRIN2B Q13224 1/20 0.44
MAPK1 P28482 1/20 0.44
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
SLC18A3 Q16572 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
CCR5 P51681 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499829 1.00 BACE1 (0.48) BACE1HTR2BNAMPTCYP19A1GRIN2B
SCHEMBL6533127 1.00 BACE1 (0.48) BACE1HTR2BNAMPTCYP19A1GRIN2B
SCHEMBL6493038 0.90 BACE1 (0.46) BACE1HTR2BNAMPTGRIN2BMAPK1
SCHEMBL6491036 0.89 GRIN2B (0.55) BACE1HTR2BNAMPTGRIN2BKCNH2
SCHEMBL6493917 0.82 RAB9A (0.46) NAMPTSLC18A3SMN1; SMN2NPC1RAB9A
SCHEMBL6492368 0.81 GRIN2B (0.56) BACE1HTR2BNAMPTGRIN2BKCNH2
SCHEMBL6490186 0.80 HTR2B (0.43) BACE1HTR2BNAMPTKCNH2HRH3
SCHEMBL19988362 0.80 HTR2B (0.64) BACE1HTR2BNAMPTKCNH2HRH3
SCHEMBL6499625 0.78 SPR (0.43) BACE1HTR2BMAPK1KCNH2HRH3
SCHEMBL6490937 0.78 BACE1 (0.43) BACE1HTR2BMAPK1KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6969724-B2 Compounds SMITHKLINE BEECHAM-SPA (GB) 2005-11-29 US disclosed