SCHEMBL6495573

SCHEMBL6495573

COC(OC)c1ccc(F)c(CN)c1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.34
AOC3 Q16853 3/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
PTGDR Q13258 1/20 0.32
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
LOXL2 Q9Y4K0 1/20 0.32
DPP8 Q6V1X1 1/20 0.31
TAAR1 Q96RJ0 2/20 0.31
IDO1 P14902 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499247 0.82 MAPK1 (0.35) DPP4CYP2D6
SCHEMBL13091292 0.79 HTR1D (0.42) DPP4CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL20256735 0.77 DPP4 (0.38) DPP4CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL2867341 0.72 PARP1 (0.37) DPP4CYP2D6IDO1PARP1
SCHEMBL6097165 0.72 ALDH1A1 (0.45) AOC3CYP3A4
SCHEMBL3536393 0.72 TAAR1 (0.55) PTGDRTAAR1IDO1
SCHEMBL27911941 0.71 DPP4 (0.41) DPP4CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL27911944 0.71 DPP4 (0.41) DPP4CYP3A4CYP2D6SLC6A2SLC6A4
SCHEMBL20256892 0.69 MAOB (0.40) PTGDRPARP1
SCHEMBL583371 0.69 TAAR1 (0.52) CYP3A4SLC6A2SLC6A4SLC6A3LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed