SCHEMBL6499247

SCHEMBL6499247

COC(OC)c1ccc(F)c(CO)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
MAP2K4 P45985 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
MAPKAPK3 Q16644 1/20 0.35
MAPK6 Q16659 1/20 0.35
GCGR P47871 1/20 0.33
DPP4 P27487 2/20 0.33
ADRB2 P07550 2/20 0.33
ADRB1 P08588 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
HIF1A Q16665 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRB3 P13945 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6495573 0.82 DPP4 (0.34) DPP4CYP2D6
SCHEMBL11994355 0.79 GCGR (0.41) MAPK1MAP2K4MAPKAPK2MAPKAPK3MAPK6
SCHEMBL19634004 0.77 MRGPRX4 (0.36) MAPK1MAP2K4MAPKAPK2MAPKAPK3MAPK6
SCHEMBL5554888 0.72 ELANE (0.49)
SCHEMBL31134127 0.72 SHBG (0.51) ADRB1TSHRNFKB1HIF1AADRA2A
SCHEMBL22709533 0.72 SHBG (0.51) ADRB1TSHRNFKB1HIF1AADRA2A
SCHEMBL2867341 0.72 PARP1 (0.37) DPP4CYP1A2CYP2D6TSHR
SCHEMBL697670 0.72 CHRM2 (0.50)
SCHEMBL2938648 0.69 LTA4H (0.39) CYP1A2CYP2D6TSHR
SCHEMBL268243 0.69 MAPK1 (0.54) MAPK1MAP2K4MAPKAPK2MAPKAPK3MAPK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed