SCHEMBL6496997

SCHEMBL6496997

CCOC(=O)C1CCN(C(=O)/C=C/c2ccc(SC)c(Cl)c2Cl)CC1

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.59
SMN1; SMN2 Q16637 6/20 0.59
NPC1 O15118 4/20 0.59
RAB9A P51151 4/20 0.59
GAA P10253 1/20 0.56
ITGB2 P05107 5/20 0.55
ICAM1 P05362 5/20 0.55
ITGAL P20701 5/20 0.55
ENPP2 Q13822 1/20 0.54
ALDH1A1 P00352 3/20 0.52
HPGD P15428 1/20 0.52
POLB P06746 1/20 0.52
HTT P42858 1/20 0.48
TSHR P16473 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6496998 1.00 KDM4E (0.59) KDM4ESMN1; SMN2NPC1RAB9AGAA
SCHEMBL6318331 0.85 ITGAL (0.62) KDM4ESMN1; SMN2NPC1RAB9AGAA
SCHEMBL6495883 0.85 ITGAL (0.68) SMN1; SMN2NPC1RAB9AITGB2ICAM1
SCHEMBL6495878 0.85 ITGAL (0.68) SMN1; SMN2NPC1RAB9AITGB2ICAM1
SCHEMBL8298709 0.85 ITGAL (0.57) KDM4ESMN1; SMN2NPC1RAB9AITGB2
SCHEMBL8298631 0.84 ITGAL (0.56) KDM4ESMN1; SMN2NPC1RAB9AITGB2
SCHEMBL6196469 0.84 ITGAL (0.78) KDM4ESMN1; SMN2NPC1RAB9AGAA
SCHEMBL6315913 0.83 ITGAL (0.54) KDM4ESMN1; SMN2NPC1RAB9AGAA
SCHEMBL6567825 0.83 ITGAL (0.54) KDM4ESMN1; SMN2NPC1RAB9AGAA
SCHEMBL6199004 0.82 ITGAL (0.77) KDM4ESMN1; SMN2NPC1RAB9AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed