SCHEMBL6497446

SCHEMBL6497446

O=C(O)/C=C/c1ccc(C(=O)OCc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.65
SLC6A2 P23975 1/20 0.65
SLC6A3 Q01959 1/20 0.65
TDP1 Q9NUW8 1/20 0.65
LMNA P02545 3/20 0.64
AKR1B10 O60218 3/20 0.60
AKR1B1 P15121 3/20 0.60
CA12 O43570 2/20 0.60
CA4 P22748 2/20 0.60
CA6 P23280 2/20 0.60
CA5A P35218 2/20 0.60
CA7 P43166 2/20 0.60
CA9 Q16790 2/20 0.60
CA14 Q9ULX7 2/20 0.60
CA5B Q9Y2D0 2/20 0.60
ALDH1A1 P00352 2/20 0.56
MAPT P10636 1/20 0.56
HPGD P15428 1/20 0.56
HCAR2 Q8TDS4 3/20 0.55
HDAC3 O15379 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6497449 1.00 KMT2A (0.65) KMT2ASLC6A2SLC6A3TDP1LMNA
SCHEMBL3089734 0.91 KMT2A (0.73) KMT2ASLC6A2SLC6A3TDP1LMNA
SCHEMBL3089736 0.91 KMT2A (0.73) KMT2ASLC6A2SLC6A3TDP1LMNA
SCHEMBL7312618 0.85 THRB (0.66) KMT2ALMNAALDH1A1MAPTHDAC3
SCHEMBL7312615 0.85 THRB (0.66) KMT2ALMNAALDH1A1MAPTHDAC3
SCHEMBL22071063 0.84 LMNA (0.84) LMNAAKR1B10AKR1B1CA12CA4
SCHEMBL312287 0.83 KMT2A (0.92) KMT2ASLC6A2SLC6A3TDP1LMNA
SCHEMBL380997 0.83 KMT2A (0.71) KMT2ASLC6A2SLC6A3TDP1LMNA
SCHEMBL25770022 0.82 MAPT (0.56) KMT2ASLC6A2SLC6A3TDP1LMNA
Benzyl Cinnamate SCHEMBL30513717 0.81 LMNA (0.90) LMNAAKR1B10AKR1B1CA12CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900318-B1 1,4,5,6-tetrahydropyrimidine derivative as a vitronectin inhibitor AVENTIS PHARMA DEUTSCLAND GMBH (DE) 2005-05-31 US disclosed
EP-1204646-B1 1,4,5,6 -TETRAHYDROPYRIMIDINE DERIVATIVE AS A VITRONECTIN INHIBITOR AVENTIS PHARMA GMBH (DE) 2004-12-29 EP disclosed
EP-1204646-A1 1,4,5,6 -TETRAHYDROPYRIMIDINE DERIVATIVE AS A VITRONECTIN INHIBITOR Aventis Pharma Deutschland GmbH (DE) 2002-05-15 EP disclosed
WO-2001007417-A1 1,4,5,6-TETRAHYDROPYRIMIDINE DERIVATIVE AS A VITRONECTIN INHIBITOR AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-02-01 WO disclosed
EP-1070707-A1 1,4,5,6-tetrahydropyrimidine derivative as a vitronectin inhibitor Aventis Pharma Deutschland GmbH (DE) 2001-01-24 EP disclosed