SCHEMBL6498941

SCHEMBL6498941

N#Cc1cccc(C2CCN(C(=O)c3cncc(CCc4ccccc4)c3)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.52
DRD3 P35462 2/20 0.52
SCD5 Q86SK9 3/20 0.46
SCD O00767 1/20 0.44
EGLN1 Q9GZT9 1/20 0.43
PARP1 P09874 1/20 0.43
MGLL Q99685 1/20 0.43
ADORA2A P29274 1/20 0.42
USP30 Q70CQ3 1/20 0.42
FASN P49327 1/20 0.41
NR3C1 P04150 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
CCR5 P51681 1/20 0.41
PARP14 Q460N5 1/20 0.41
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1871107 0.85 GRM5 (0.48) DRD2DRD3SCD5SCDEGLN1
SCHEMBL7021172 0.85 TPSAB1 (0.53)
SCHEMBL7018734 0.84 TPSAB1 (0.46) PARP1NPC1RAB9ACCR5PARP14
Hydrochloric Acid SCHEMBL4402047 0.84 TPSAB1 (0.52)
SCHEMBL1872130 0.83 HPN (0.47) PARP1NPC1RAB9ACCR5PARP14
SCHEMBL1870287 0.82 CHRM4 (0.48) DRD2PARP1
Hydrochloric Acid SCHEMBL1867557 0.82 HPN (0.46) PARP1NPC1RAB9ACCR5PARP14
SCHEMBL6501829 0.81 TPSAB1 (0.42) PARP1MGLLNPC1RAB9ACCR5
SCHEMBL6498937 0.81 FASN (0.46) DRD2DRD3SCD5SCDMGLL
Hydrochloric Acid SCHEMBL7107726 0.80 TPSAB1 (0.41) PARP1MGLLNPC1RAB9ACCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6977263-B2 Chemical compounds AVENTIS PHARMACEUTICALS INC. (US) 2005-12-20 US disclosed