SCHEMBL7018734

SCHEMBL7018734

NCCc1cccc(C2CCN(C(=O)c3cncc(CCc4ccccc4)c3)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 7/20 0.46
PARP1 P09874 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CCR5 P51681 1/20 0.42
PARP14 Q460N5 1/20 0.42
PARP10 Q53GL7 1/20 0.42
F10 P00742 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7021172 0.93 TPSAB1 (0.53) TPSAB1F10
Hydrochloric Acid SCHEMBL4402047 0.92 TPSAB1 (0.52) TPSAB1F10
SCHEMBL7027368 0.88 TPSAB1 (0.45) TPSAB1CA12CA1CA2CA7
Hydrochloric Acid SCHEMBL4395982 0.87 TPSAB1 (0.44) TPSAB1CA12CA1CA2CA7
SCHEMBL1872130 0.86 HPN (0.47) PARP1CA12CA1CA2CA7
Hydrochloric Acid SCHEMBL1867557 0.85 HPN (0.46) PARP1CA12CA1CA2CA7
SCHEMBL6501829 0.85 TPSAB1 (0.42) TPSAB1PARP1CA12CA1CA2
SCHEMBL7025350 0.84 TPSAB1 (0.42) TPSAB1PARP1CA12CA1CA2
SCHEMBL6498941 0.84 DRD2 (0.52) PARP1NPC1RAB9ACCR5PARP14
Hydrochloric Acid SCHEMBL7107726 0.84 TPSAB1 (0.41) TPSAB1PARP1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS Aventis Pharmaceuticals Inc. (US) 2003-04-02 EP disclosed
WO-2001090101-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2001-11-29 WO disclosed