SCHEMBL6499308

SCHEMBL6499308

[c]1cc2ccccc2nc1-c1cnc2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 4/20 0.51
PDGFRA P16234 4/20 0.51
CYP2A6 P11509 1/20 0.49
BIRC5 O15392 1/20 0.47
PIK3CD O00329 2/20 0.46
PIK3CA P42336 2/20 0.46
CYP1A2 P05177 1/20 0.44
NISCH Q9Y2I1 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
MAP4K4 O95819 1/20 0.42
CSNK1G2 P78368 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
MAP4K5 Q9Y4K4 1/20 0.42
TOP2A P11388 1/20 0.42
TOP2B Q02880 1/20 0.42
ALDH1A1 P00352 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3986805 0.83 NPC1 (0.59) PDGFRBPDGFRACYP2A6PIK3CDPIK3CA
SCHEMBL8637618 0.79 GSTP1 (0.40) CYP1A2ALDH1A1MAPTNPC1RAB9A
SCHEMBL2996550 0.78 PDE10A (0.40) CYP1A2CA12CA9ALDH1A1MAPT
SCHEMBL32667946 0.78 PDGFRB (0.77) PDGFRBPDGFRACYP2A6BIRC5PIK3CD
SCHEMBL2772360 0.78 PDGFRB (0.77) PDGFRBPDGFRACYP2A6BIRC5PIK3CD
SCHEMBL16720404 0.75 ADORA2A (0.43) PDGFRBPDGFRAMAP4K4ALDH1A1MAPT
SCHEMBL7873327 0.75 PDGFRB (0.54) PDGFRBPDGFRACYP2A6BIRC5PIK3CD
SCHEMBL16720376 0.74 NPC1 (0.50) PDGFRBPDGFRACYP1A2ALDH1A1MAPT
SCHEMBL12504960 0.72 AR (0.51) ALDH1A1MAPTNPC1RAB9AGLA
SCHEMBL708999 0.72 PDGFRB (0.75) PDGFRBPDGFRACYP2A6BIRC5PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed
US-6127386-A STIMULANTS, NEUROTRANSMITTERS, CHOLINERGIC AGENTS ABBOTT LABORATORIES (US) 2000-10-03 US disclosed
EP-0797786-A4 INCORPORATING PHOTOCHROMIC MOLECULES IN LIGHT TRANSMISSIBLE ARTICLES SOLA INT HOLDINGS (AU) 1998-12-09 EP disclosed
EP-0797786-A1 INCORPORATING PHOTOCHROMIC MOLECULES IN LIGHT TRANSMISSIBLE ARTICLES SOLA INTERNATIONAL HOLDINGS, LTD. (AU) 1997-10-01 EP disclosed
WO-1996018928-A1 INCORPORATING PHOTOCHROMIC MOLECULES IN LIGHT TRANSMISSIBLE ARTICLES SOLA INTERNATIONAL HOLDINGS LTD. (AU) 1996-06-20 WO disclosed