SCHEMBL6499398

SCHEMBL6499398

CC(NC(=O)C1CCN(C(=O)C=Cc2cc3c(cc2Cl)OCO3)CC1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MAOB P27338 2/20 0.44
POLB P06746 1/20 0.43
CAPN1 P07384 3/20 0.41
ITGAL P20701 5/20 0.41
ITGB2 P05107 3/20 0.41
ICAM1 P05362 3/20 0.41
MAPT P10636 2/20 0.40
USP2 O75604 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
GAA P10253 1/20 0.40
GABRA1 P14867 1/20 0.40
GABRB2 P47870 1/20 0.40
HPGD P15428 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6532940 1.00 NPC1 (0.47) NPC1RAB9AMAOBPOLBCAPN1
SCHEMBL6497505 0.89 NPC1 (0.47) NPC1RAB9AMAOBPOLBCAPN1
SCHEMBL6503994 0.83 CAPN1 (0.45) NPC1RAB9ACAPN1ITGALITGB2
SCHEMBL6497738 0.83 RAB9A (0.53) NPC1RAB9ACAPN1ITGALITGB2
SCHEMBL6497734 0.83 RAB9A (0.53) NPC1RAB9ACAPN1ITGALITGB2
SCHEMBL6503990 0.83 CAPN1 (0.45) NPC1RAB9ACAPN1ITGALITGB2
SCHEMBL6503421 0.82 ITGAL (0.48) NPC1RAB9APOLBCAPN1ITGAL
SCHEMBL8296029 0.82 ITGAL (0.48) NPC1RAB9APOLBCAPN1ITGAL
SCHEMBL6503425 0.82 ITGAL (0.48) NPC1RAB9APOLBCAPN1ITGAL
SCHEMBL6497639 0.82 CAPN1 (0.42) NPC1RAB9APOLBCAPN1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed