SCHEMBL6500228

SCHEMBL6500228

CSc1ccc(C=CC(=O)N2CCC(C(=O)N[C@@H](CNC(=O)c3cccc(Cl)c3)C(=O)O)CC2)c(Cl)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 10/20 0.46
ITGB2 P05107 9/20 0.46
ICAM1 P05362 9/20 0.46
CAPN1 P07384 4/20 0.41
CASP3 P42574 1/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6500234 1.00 ITGAL (0.46) ITGALITGB2ICAM1CAPN1CASP3
SCHEMBL6495913 0.93 ITGAL (0.51) ITGALITGB2ICAM1CAPN1MEN1
SCHEMBL6495908 0.93 ITGAL (0.51) ITGALITGB2ICAM1CAPN1MEN1
SCHEMBL8297366 0.93 ITGAL (0.51) ITGALITGB2ICAM1CAPN1MEN1
SCHEMBL6498508 0.93 ITGAL (0.45) ITGALITGB2ICAM1CAPN1CASP3
SCHEMBL6498494 0.93 ITGAL (0.45) ITGALITGB2ICAM1CAPN1CASP3
SCHEMBL6498498 0.93 ITGAL (0.45) ITGALITGB2ICAM1CAPN1CASP3
SCHEMBL6503350 0.92 ITGAL (0.44) ITGALITGB2ICAM1CAPN1MEN1
SCHEMBL6500717 0.92 ITGAL (0.47) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6500735 0.92 ITGAL (0.47) ITGALITGB2ICAM1CAPN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed