SCHEMBL6501803

SCHEMBL6501803

COc1ccc(-n2cc(C(=O)NN)nc2-c2ccc(Cl)cc2Cl)cc1

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 18/20 0.72
CNR2 P34972 5/20 0.58
GABRA2 P47869 1/20 0.50
GABRB2 P47870 1/20 0.50
MARS1 P56192 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6343454 0.88 CNR1 (0.67) CNR1CNR2GABRA2GABRB2MARS1
SCHEMBL6332950 0.87 CNR1 (0.68) CNR1CNR2GABRA2GABRB2MARS1
SCHEMBL4507104 0.84 CNR1 (0.84) CNR1CNR2
SCHEMBL5370038 0.84 CNR1 (0.62) CNR1CNR2GABRA2GABRB2
SCHEMBL4516531 0.84 CNR1 (1.00) CNR1CNR2
SCHEMBL6343712 0.83 CNR1 (0.61) CNR1CNR2
SCHEMBL6334842 0.83 CNR1 (0.61) CNR1CNR2
SCHEMBL4510717 0.82 CNR1 (0.65) CNR1CNR2
SCHEMBL6334651 0.81 CNR1 (0.85) CNR1CNR2
SCHEMBL6334654 0.81 CNR1 (0.85) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050256167-A1 Preparation and use of imidazole derivatives for treatment of obesity BAYER PHARMACEUTICALS CORPORATION (US) 2005-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050256167-A1 Preparation and use of imidazole derivatives for treatment of obesity GPR119, GIPR, PGC CNR1 405/4885CNR2 340/4885GABRA2 981/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.