SCHEMBL6501838

SCHEMBL6501838

O=CNc1nc(-c2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 3/20 0.58
MAPT P10636 3/20 0.58
TDP1 Q9NUW8 1/20 0.58
ADORA1 P30542 12/20 0.54
ADORA3 P0DMS8 5/20 0.54
ADORA2A P29274 4/20 0.50
ADORA2B P29275 1/20 0.50
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6508924 0.83 ADORA1 (0.82) MAPTADORA1ADORA3ADORA2AADORA2B
SCHEMBL4829403 0.77 ADORA1 (0.58) ADORA1ADORA3ADORA2AADORA2BMEN1
SCHEMBL23969914 0.75 ALDH1A1 (0.52) AGTR1MAPTTDP1ADORA1ADORA3
SCHEMBL12496376 0.74 ALDH1A1 (0.41) MAPTADORA1MEN1ALDH1A1HPGD
SCHEMBL28193696 0.74 SLC2A1 (0.56) SMN1; SMN2KDM4E
SCHEMBL26523872 0.74 TDP1 (1.00) AGTR1MAPTTDP1ADORA1ADORA3
SCHEMBL2401750 0.74 MAPT (1.00) AGTR1MAPTTDP1ADORA1ADORA3
SCHEMBL6529699 0.73 ADORA1 (0.74) AGTR1MAPTTDP1ADORA1ADORA3
SCHEMBL15871200 0.72 MAPT (0.62) AGTR1MAPTTDP1ADORA1ADORA3
SCHEMBL49700 0.72 ADORA2A (0.58) ADORA1ADORA3ADORA2AADORA2BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO claimed
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO disclosed