SCHEMBL6503528

SCHEMBL6503528

COC(=O)[C@H](Cc1ccc(-c2ccccc2)c(Oc2ccccc2)c1)NC(=O)c1cc(Cl)ccc1N

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PYGL P06737 1/20 0.46
PSMB5 P28074 4/20 0.44
LNPEP Q9UIQ6 1/20 0.44
TACR3 P29371 1/20 0.43
CDK2 P24941 3/20 0.42
TSHR P16473 1/20 0.42
FNTA P49354 1/20 0.42
FNTB P49356 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
NOS2 P35228 1/20 0.41
CTNNB1 P35222 1/20 0.41
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6503531 1.00 PYGL (0.46) PYGLPSMB5LNPEPTACR3CDK2
SCHEMBL3971232 0.93 PYGL (0.47) PYGLPSMB5LNPEPTACR3CDK2
SCHEMBL3979419 0.93 PYGL (0.47) PYGLPSMB5LNPEPTACR3CDK2
SCHEMBL3974514 0.89 PYGL (0.50) PYGLLNPEPTACR3CDK2TSHR
SCHEMBL3974510 0.89 PYGL (0.50) PYGLLNPEPTACR3CDK2TSHR
SCHEMBL5926278 0.86 PYGL (0.55) PYGLPSMB5LNPEPTACR3CDK2
SCHEMBL3991444 0.84 ITGA4 (0.48)
SCHEMBL5927011 0.84 ITGA4 (0.48)
SCHEMBL3998558 0.83 ABCG2 (0.48) LNPEPTACR3TSHRKDM4EALDH1A1
SCHEMBL3996954 0.83 ABCG2 (0.48) LNPEPTACR3TSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005014532-A1 ARYL AND HETEROARYL COMPOUNDS, COMPOSITIONS AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2005-02-17 WO disclosed