SCHEMBL6505155

SCHEMBL6505155

COc1cc2c(c(OC)c1)C(c1ccc(O)cc1)N(C(=O)c1cccs1)CC2

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2C Q14957 4/20 0.53
HSD17B10 Q99714 1/20 0.50
FKBP1A P62942 1/20 0.49
GAA P10253 2/20 0.48
LMNA P02545 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HPGD P15428 1/20 0.47
MTNR1B P49286 1/20 0.45
CYP3A4 P08684 1/20 0.44
MAPK1 P28482 1/20 0.44
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
SIRT5 Q9NXA8 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
NPC1 O15118 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13972856 1.00 GRIN2C (0.53) GRIN2CHSD17B10FKBP1AGAALMNA
SCHEMBL4414980 0.83 KMT2A (0.60) GRIN2CFKBP1ALMNAMTNR1BMEN1
SCHEMBL4423041 0.82 GRIN2C (0.54) GRIN2CMTNR1BMEN1KMT2A
SCHEMBL4423052 0.81 GRIN2C (0.57) GRIN2CLMNAMTNR1BMEN1KMT2A
SCHEMBL4421006 0.80 ABCG2 (0.51) GRIN2CMTNR1BMEN1KMT2A
SCHEMBL4422963 0.79 GRIN2C (0.47) GRIN2CFKBP1AGAALMNAMTNR1B
SCHEMBL4416765 0.79 KMT2A (0.51) GRIN2CLMNAMTNR1BMEN1KMT2A
SCHEMBL4416816 0.78 GRIN2C (0.44) GRIN2CGAALMNAHPGDMTNR1B
SCHEMBL4425728 0.78 GRIN2C (0.43) GRIN2CSMN1; SMN2HPGDMTNR1BMAPK1
SCHEMBL4413283 0.78 MTNR1B (0.46) GRIN2CFKBP1AMTNR1BMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050070570-A1 Novel potassium channels modulators 4SC AG (DE) 2005-03-31 US disclosed
EP-1489071-A1 N-substituted, 3,4-dihydro-1H-isoquinoline as potassium channels modulators 4SC AG (DE) 2004-12-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050070570-A1 Novel potassium channels modulators HCN4, KCNA4, KCNN4 GRIN2C 567/4885HSD17B10 1517/4885FKBP1A 3805/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.