SCHEMBL4607220

SCHEMBL4607220

CC(O)C(NC1CC1)Oc1cccc2[nH]c3ccccc3c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 9/20 0.48
ADRB2 P07550 10/20 0.48
DNM1 Q05193 2/20 0.48
ADRB1 P08588 5/20 0.41
UTS2R Q9UKP6 1/20 0.41
TLR4 O00206 4/20 0.41
DRD2 P14416 3/20 0.41
KDM4E B2RXH2 1/20 0.41
SLC22A2 O15244 1/20 0.41
SLC22A1 O15245 1/20 0.41
MLNR O43193 1/20 0.41
NR1I2 O75469 1/20 0.41
KCNK2 O95069 1/20 0.41
ABCB11 O95342 1/20 0.41
APP P05067 1/20 0.41
ABCB1 P08183 1/20 0.41
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4795725 0.95 ADRB2 (0.49) ADRB3ADRB2DNM1ADRB1TLR4
SCHEMBL4643608 0.93 ADRB3 (0.46) ADRB3ADRB2DNM1ADRB1TLR4
SCHEMBL4607115 0.86 ADRB3 (0.50) ADRB3ADRB2DNM1ADRB1HTR2A
SCHEMBL4608341 0.84 ADRB2 (0.53) ADRB3ADRB2DNM1ADRB1TLR4
SCHEMBL9621537 0.83 ADRB2 (0.55) ADRB3ADRB2DNM1ADRB1TLR4
SCHEMBL4727264 0.81 ADRB2 (0.50) ADRB3ADRB2DNM1ADRB1TLR4
SCHEMBL6507182 0.79 ADRB2 (0.54) ADRB3ADRB2DNM1ADRB1UTS2R
SCHEMBL4696496 0.79 ALDH1A1 (0.41) ADRB3ADRB2ADRB1MAPTKMT2A
SCHEMBL7701306 0.78 ADRB3 (0.68) ADRB3ADRB2DNM1ADRB1UTS2R
SCHEMBL4457452 0.78 ADRB2 (0.53) ADRB3ADRB2DNM1ADRB1UTS2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed