SCHEMBL6507791

SCHEMBL6507791

O=C(NC1CCCCC1)c1c(CN2CCC(N3CCCCC3)CC2)c(-c2ccccc2)nc2ncccc12

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 8/20 0.62
TACR2 P21452 7/20 0.62
OPRM1 P35372 4/20 0.62
TRPV4 Q9HBA0 13/20 0.58
KCNH2 Q12809 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5945397 0.89 TACR3 (0.77) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL6506812 0.87 TRPV4 (0.58) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL5732536 0.81 TACR2 (0.71) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL7225413 0.76 TRPV4 (0.67) TACR3TACR2OPRM1TRPV4
SCHEMBL5945344 0.76 TRPV4 (0.80) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL2373330 0.76 TRPV4 (0.72) TACR3TACR2OPRM1TRPV4KCNH2
Hydrochloric Acid SCHEMBL5733490 0.75 TRPV4 (0.71) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL6533888 0.75 TRPV4 (0.54) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL5203642 0.75 TRPV4 (0.73) TACR3TACR2OPRM1TRPV4KCNH2
SCHEMBL6428018 0.74 TRPV4 (0.70) TACR3TACR2OPRM1TRPV4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016878-A2 METHODS FOR THE PREPARATION OF 5-FLUORO-PYRROLO[2,3-d]PYRIMIDINE COMPOUNDS ISIS PHARMACEUTICALS, INC. (US) 2005-02-24 WO claimed
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO claimed
CN-101531695-A Method for synthesizing fluoro-oligonucleotide for preparing siRNA ZHENGZHOU RUISAI TECHNOLOGY AN 2009-09-16 CN disclosed
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed