SCHEMBL6506812

SCHEMBL6506812

COC(=O)c1c(CN2CCC(N3CCCCC3)CC2)c(-c2ccccc2)nc2ncccc12

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 13/20 0.58
TACR3 P29371 9/20 0.58
TACR2 P21452 7/20 0.58
OPRM1 P35372 3/20 0.57
KCNH2 Q12809 3/20 0.53
CACNA1C Q13936 1/20 0.49
SCN5A Q14524 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203642 0.88 TRPV4 (0.73) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL6507791 0.87 TACR3 (0.62) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL6528864 0.86 TRPV4 (0.55) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL6853291 0.81 TRPV4 (0.55) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL5945408 0.81 TRPV4 (0.55) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL5202474 0.79 TACR3 (0.59) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL2373330 0.78 TRPV4 (0.72) TRPV4TACR3TACR2OPRM1KCNH2
Hydrochloric Acid SCHEMBL5733490 0.77 TRPV4 (0.71) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL6533888 0.77 TRPV4 (0.54) TRPV4TACR3TACR2OPRM1KCNH2
SCHEMBL4237458 0.76 TACR3 (0.88) TRPV4TACR3TACR2OPRM1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed