SCHEMBL6508630

SCHEMBL6508630

CCCCN1[CH]COCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MAPK1 P28482 2/20 0.38
CYP1A2 P05177 1/20 0.38
CHRM2 P08172 1/20 0.38
CHRM1 P11229 1/20 0.38
HTR2A P28223 1/20 0.38
SCN1A P35498 1/20 0.38
HTR2B P41595 1/20 0.38
KCNH2 Q12809 1/20 0.38
SCN2A Q99250 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
SCN3A Q9NY46 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
LMNA P02545 3/20 0.37
USP2 O75604 1/20 0.37
TSHR P16473 1/20 0.35
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTT P42858 1/20 0.32
THRB P10828 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1078460 0.94 SIGMAR1 (0.37) ALDH1A1MAPK1CYP1A2CHRM2CHRM1
SCHEMBL151371 0.88
SCHEMBL1456336 0.69 DAO (0.35) LMNASMN1; SMN2HTTKMT2A
SCHEMBL4914244 0.68
SCHEMBL84935 0.67 ALDH1A1 (0.61) ALDH1A1MAPK1CYP1A2CHRM2CHRM1
SCHEMBL2099498 0.67 CYP1A2 (0.34) CYP1A2TSHRHTTKMT2AMEN1
Pentane SCHEMBL8722577 0.66 MAPK1 (0.46) ALDH1A1MAPK1CYP1A2CHRM2CHRM1
SCHEMBL37780 0.66
Pentane SCHEMBL28256229 0.66 MAPK1 (0.46) ALDH1A1MAPK1CYP1A2CHRM2CHRM1
Hydrochloric Acid SCHEMBL25342847 0.66 MAPK1 (0.62) ALDH1A1MAPK1CYP1A2CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0810209-A2 Alpha - and beta-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors G.D. SEARLE & CO. (US) 1997-12-03 EP claimed
WO-2005021506-A1 SYNTHESIS OF 1-[4-(2-METHOXYPHENYL) PIPERAZIN-1-YL]-3-(2,6-DIOXOPIPERIDIN-1-YL) PROPANE RANBAXY LABORATORIES LIMITED (IN) 2005-03-10 WO disclosed
EP-0810209-A2 Alpha - and beta-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors G.D. SEARLE & CO. (US) 1997-12-03 EP disclosed
EP-0470514-B1 Carbostyril derivatives and pharmaceutical composition containing the same OTSUKA PHARMA CO LTD (JP) 1997-02-19 EP disclosed
US-5300513-A Vasopressin antagonists; vasodilators, hypotensive agents, water diuretics, and platelet agglutination inhibitors OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-05 US disclosed
EP-0470514-A1 Carbostyril derivatives and pharmaceutical composition containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-02-12 EP disclosed